SCHEMBL6985322

SCHEMBL6985322

N#Cc1ccc(CCC(=O)N2CCCc3cccc(NS(=O)(=O)c4ccccc4)c32)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.41
NR3C1 P04150 2/20 0.40
AR P10275 1/20 0.40
METAP2 P50579 1/20 0.39
PKM P14618 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 1/20 0.38
LSS P48449 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
THRB P10828 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
FPR1 P21462 2/20 0.37
FPR2 P25090 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7408050 0.92 TP53 (0.40) GAANR3C1PKMMEN1KMT2A
SCHEMBL6982764 0.92 FPR1 (0.43) GAANR3C1METAP2PKMMEN1
SCHEMBL6985749 0.92 ALDH1A1 (0.48) GAANR3C1PKMMEN1KMT2A
SCHEMBL6984759 0.92 LMNA (0.47) GAANR3C1PKMMEN1KMT2A
SCHEMBL6983505 0.91 NR3C1 (0.42) NR3C1ARPKMMEN1KMT2A
SCHEMBL6984039 0.91 TP53 (0.45) GAANR3C1ARPKMALDH1A1
SCHEMBL7411038 0.91 PKM (0.43) GAANR3C1ARPKMMEN1
SCHEMBL6977498 0.91 CCKBR (0.44) GAANR3C1ARPKMMEN1
SCHEMBL6982163 0.90 SLC16A3 (0.45) GAANR3C1PKMMEN1KMT2A
SCHEMBL6981583 0.90 STAT3 (0.49) GAANR3C1PKMMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed