SCHEMBL6979094

SCHEMBL6979094

CC(CC[C@H]1NC(=N)C[C@@H]1C)NCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.47
BCHE P06276 1/20 0.39
GAA P10253 1/20 0.36
ATM Q13315 1/20 0.36
LMNA P02545 1/20 0.35
POLB P06746 2/20 0.34
MAPK1 P28482 1/20 0.34
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
HTR1A P08908 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
DRD2 P14416 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
CNR1 P21554 1/20 0.33
SLC6A2 P23975 1/20 0.33
HTR2A P28223 1/20 0.33
SLC6A4 P31645 1/20 0.33
MC4R P32245 1/20 0.33
ADRA1A P35348 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6970998 1.00 SIGMAR1 (0.47) SIGMAR1BCHEGAAATMLMNA
SCHEMBL6969440 0.79 MEN1 (0.43) SIGMAR1GAAHTR2AKMT2A
Hydrochloric Acid SCHEMBL27426481 0.78 MEN1 (0.42) SIGMAR1GAAKMT2A
SCHEMBL6980288 0.77 MAOA (0.45) SIGMAR1GAAKMT2A
SCHEMBL6977437 0.77 MAOA (0.45) SIGMAR1GAAKMT2A
SCHEMBL6971448 0.73 NOS1 (0.41)
SCHEMBL6977148 0.73 NOS1 (0.41)
SCHEMBL6970605 0.69 ALDH1A1 (0.43) SIGMAR1HTR2AHRH1OPRK1
SCHEMBL10451642 0.66 BCHE (0.71) SIGMAR1BCHEGAAATMOPRK1
SCHEMBL11096038 0.66 BCHE (0.71) SIGMAR1BCHEGAAATMOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821674-B1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS SEARLE & CO (US) 2003-08-06 EP claimed
US-6011028-A Cyclic amidino agents useful as nitric oxide synthase inhibitors G.D. SEARLE & CO. (US) 2000-01-04 US claimed
EP-0821674-B1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS SEARLE & CO (US) 2003-08-06 EP disclosed
US-6011028-A Cyclic amidino agents useful as nitric oxide synthase inhibitors G.D. SEARLE & CO. (US) 2000-01-04 US disclosed