SCHEMBL6979712

SCHEMBL6979712

COC(=O)CCCN(c1ccc2c(c1)CCCN2C(=O)CCc1ccc(C(=O)OCc2ccccc2)cc1C(=N)N)S(=O)(=O)c1cccc2ccccc12

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
F2 P00734 3/20 0.35
RORC P51449 1/20 0.34
PARP1 P09874 1/20 0.34
THRB P10828 1/20 0.33
NR3C1 P04150 3/20 0.33
AVPR2 P30518 1/20 0.32
SRD5A1 P18405 1/20 0.32
SRD5A2 P31213 1/20 0.32
USP2 O75604 1/20 0.31
PKM P14618 1/20 0.31
F10 P00742 2/20 0.31
ALDH1A1 P00352 2/20 0.31
F7 P08709 1/20 0.31
MEN1 O00255 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31
PLAU P00749 1/20 0.31
NOTUM Q6P988 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6982379 0.91 THRB (0.35) F2RORCPARP1THRBNR3C1
SCHEMBL7085095 0.91 ALDH1A1 (0.36) RORCPARP1THRBNR3C1SRD5A1
SCHEMBL7089640 0.90 PDK1 (0.36) F2RORCPARP1THRBNR3C1
SCHEMBL7088164 0.89 THRB (0.36) PARP1THRBNR3C1SRD5A1SRD5A2
SCHEMBL6984290 0.88 F10 (0.35) F2RORCPARP1THRBNR3C1
SCHEMBL6981981 0.86 F2 (0.40) F2RORCPARP1NR3C1USP2
SCHEMBL6978636 0.85 PDK1 (0.36) RORCPARP1THRBNR3C1USP2
SCHEMBL6976718 0.83 NR3C1 (0.42) F2NR3C1F10ALDH1A1HPGD
SCHEMBL7084262 0.80 F2 (0.46) F2RORCPARP1NR3C1F10
SCHEMBL6984481 0.77 F2 (0.41) F2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
US-6300342-B1 FOR THERAPY OR INHIBITING THROMBUS FORMATION; FOR THERAPY OF FIBRIN-DEPENDENT INFLAMMATORY CONDITION BOEHRINGER INGELHEIM PHARM KG (DE) 2001-10-09 US disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed