SCHEMBL6982379

SCHEMBL6982379

CCOC(=O)CCN(c1ccc2c(c1)CCCN2C(=O)CCc1ccc(C(=O)OCc2ccccc2)cc1C(=N)N)S(=O)(=O)c1cccc2ccccc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.35
GAA P10253 1/20 0.35
PARP1 P09874 1/20 0.34
ALDH1A1 P00352 3/20 0.34
HPGD P15428 2/20 0.34
LMNA P02545 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
SRD5A1 P18405 1/20 0.33
SRD5A2 P31213 1/20 0.33
POLB P06746 1/20 0.33
RORC P51449 1/20 0.33
NR3C1 P04150 2/20 0.33
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NOTUM Q6P988 2/20 0.33
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7089640 0.95 PDK1 (0.36) THRBPARP1ALDH1A1HPGDLMNA
SCHEMBL6979712 0.91 F2 (0.35) THRBPARP1ALDH1A1HPGDSRD5A1
SCHEMBL7085095 0.91 ALDH1A1 (0.36) THRBPARP1ALDH1A1HPGDLMNA
SCHEMBL6978636 0.90 PDK1 (0.36) THRBPARP1ALDH1A1HPGDLMNA
SCHEMBL6984290 0.90 F10 (0.35) THRBPARP1ALDH1A1SRD5A1SRD5A2
SCHEMBL7088164 0.89 THRB (0.36) THRBPARP1ALDH1A1HPGDLMNA
SCHEMBL6976718 0.82 NR3C1 (0.42) ALDH1A1HPGDLMNANPSR1NR3C1
Hydrochloric Acid SCHEMBL6979622 0.81 F2 (0.39) PARP1ALDH1A1POLBRORCNR3C1
SCHEMBL6984481 0.80 F2 (0.41) GAAALDH1A1HPGDLMNANPSR1
SCHEMBL6979175 0.79 USP2 (0.39) GAAALDH1A1HPGDLMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
US-6300342-B1 FOR THERAPY OR INHIBITING THROMBUS FORMATION; FOR THERAPY OF FIBRIN-DEPENDENT INFLAMMATORY CONDITION BOEHRINGER INGELHEIM PHARM KG (DE) 2001-10-09 US disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed