SCHEMBL6979787

SCHEMBL6979787

CCOC(=O)Cc1ccccc1S(=O)(=O)Nc1ccc2c(c1)CCCN2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.39
HIF1A Q16665 3/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
CREBBP Q92793 2/20 0.38
AURKA O14965 2/20 0.37
AURKB Q96GD4 2/20 0.37
POLB P06746 2/20 0.37
TRIM24 O15164 1/20 0.37
KDM4E B2RXH2 2/20 0.37
NR3C1 P04150 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6980011 0.79 BRD4 (0.58) BRD4CREBBPPOLBMAPTALDH1A1
SCHEMBL6985547 0.78 HTR6 (0.41) BRD4HDAC3HDAC4HDAC1HDAC7
SCHEMBL6983879 0.74 ALDH1A1 (0.53) POLBKDM4EMAPTALDH1A1PKM
SCHEMBL8768330 0.73 MAPT (0.49) KDM4EMAPTALDH1A1PKMLMNA
SCHEMBL6983095 0.73 BRD4 (0.51) BRD4HDAC1ALDH1A1TSHR
SCHEMBL6987762 0.73 BRD4 (0.48) BRD4CREBBPTRIM24NR3C1MAPT
SCHEMBL6984820 0.72 HTR6 (0.61) BRD4KDM4EMAPTALDH1A1PKM
SCHEMBL6985107 0.70 LMNA (0.67) BRD4POLBMAPTALDH1A1PKM
SCHEMBL6982230 0.70 NR3C1 (0.47) BRD4CREBBPTRIM24NR3C1MAPT
SCHEMBL14815944 0.69 HRH3 (0.49) POLBKDM4EMAPTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed