SCHEMBL6980097

SCHEMBL6980097

CCCN(CCC)C(=O)CN(Cc1ccccc1)c1cccc2c1N(C(=O)CCc1ccc(C#N)cc1)CCC2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.37
RORC P51449 1/20 0.37
AVPR2 P30518 2/20 0.34
OXTR P30559 2/20 0.34
AVPR1A P37288 2/20 0.34
ALDH1A1 P00352 3/20 0.34
TSHR P16473 3/20 0.34
KDM4E B2RXH2 2/20 0.34
LMNA P02545 1/20 0.34
NPC1 O15118 2/20 0.33
MAPT P10636 2/20 0.33
MAPK1 P28482 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MEP1B Q16820 1/20 0.33
TP53 P04637 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
TMEM97 Q5BJF2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6979172 0.89 KDM1A (0.41) KDM1AALDH1A1TSHRKDM4ENPC1
SCHEMBL6982692 0.88 L3MBTL1 (0.38) KDM1AALDH1A1TSHRKDM4ELMNA
SCHEMBL6984169 0.88 KDM1A (0.38) KDM1ARORCAVPR2OXTRAVPR1A
SCHEMBL7090381 0.86 TP53 (0.38) KDM1ARORCALDH1A1TSHRKDM4E
SCHEMBL6977076 0.86 RORC (0.41) KDM1ARORCALDH1A1MAPTSMN1; SMN2
SCHEMBL6980094 0.85 KDM1A (0.42) KDM1ARORCALDH1A1TSHRLMNA
SCHEMBL6986002 0.84 RXRA (0.45) KDM1ARORCALDH1A1TSHRKDM4E
SCHEMBL6981595 0.83 LTB4R2 (0.46) AVPR2OXTRAVPR1AALDH1A1TSHR
SCHEMBL6986008 0.83 MEN1 (0.39) RORCAVPR2OXTRAVPR1AALDH1A1
SCHEMBL6987632 0.81 ALDH1A1 (0.39) RORCALDH1A1TSHRLMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed