SCHEMBL6980541

SCHEMBL6980541

N#Cc1ccc(OCC(=O)N2CCCc3cccc(NS(=O)(=O)c4ccccc4)c32)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.48
GAA P10253 1/20 0.48
CTDSP1 Q9GZU7 1/20 0.43
ALDH1A1 P00352 3/20 0.42
AR P10275 2/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
USP2 O75604 1/20 0.41
LMNA P02545 1/20 0.41
ALOX15 P16050 1/20 0.41
TUBB4A P04350 1/20 0.41
TUBB P07437 1/20 0.41
TUBA3C P0DPH7 1/20 0.41
TUBA1B P68363 1/20 0.41
TUBA4A P68366 1/20 0.41
TUBB4B P68371 1/20 0.41
TUBB3 Q13509 1/20 0.41
TUBB2A Q13885 1/20 0.41
TUBB8 Q3ZCM7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985835 0.87 SLC16A3 (0.42) HSD17B10GAAALDH1A1MEN1KMT2A
SCHEMBL6985322 0.86 GAA (0.41) GAAALDH1A1ARMEN1KMT2A
SCHEMBL6985371 0.84 NR3C1 (0.44) GAAALDH1A1ARLMNAPKM
SCHEMBL6976883 0.83 NR3C1 (0.38) ALDH1A1ARMEN1KMT2ASMN1; SMN2
SCHEMBL7406048 0.83 EEF2K (0.39) HSD17B10ALDH1A1ARMEN1KMT2A
SCHEMBL6982980 0.83 PKM (0.39) HSD17B10ALDH1A1ARMEN1KMT2A
SCHEMBL6983048 0.82 NAMPT (0.41) ALDH1A1ARMEN1KMT2ALMNA
SCHEMBL6980538 0.82 NR3C1 (0.56) ALDH1A1ARSMN1; SMN2LMNAMAPT
SCHEMBL6981583 0.81 STAT3 (0.49) GAAALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL6983505 0.81 NR3C1 (0.42) HSD17B10ALDH1A1ARMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed