SCHEMBL6985371

SCHEMBL6985371

N#Cc1ccc(C(=O)N2CCCc3cccc(NS(=O)(=O)c4ccccc4)c32)cc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 2/20 0.44
AR P10275 1/20 0.44
SLC16A3 O15427 1/20 0.44
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 2/20 0.42
LMNA P02545 1/20 0.42
MAPK1 P28482 1/20 0.42
SLC22A12 Q96S37 1/20 0.42
HTT P42858 1/20 0.41
PKM P14618 1/20 0.41
GAA P10253 1/20 0.40
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983048 0.84 NAMPT (0.41) NR3C1ARALDH1A1LMNAHTT
SCHEMBL6984554 0.84 ALDH1A1 (0.44) NR3C1ARSLC16A3L3MBTL1ALDH1A1
SCHEMBL6980541 0.84 HSD17B10 (0.48) NR3C1ARALDH1A1LMNAHTT
SCHEMBL6985322 0.84 GAA (0.41) NR3C1ARALDH1A1LMNAPKM
SCHEMBL6981761 0.82 LIMK2 (0.40) NR3C1ARALDH1A1LMNAPKM
SCHEMBL7406048 0.82 EEF2K (0.39) NR3C1ARSLC16A3ALDH1A1LMNA
SCHEMBL6982980 0.82 PKM (0.39) NR3C1ARALDH1A1LMNASLC22A12
SCHEMBL6976883 0.82 NR3C1 (0.38) NR3C1ARALDH1A1LMNASLC22A12
SCHEMBL6985366 0.80 NR3C1 (0.66) NR3C1ALDH1A1LMNA
SCHEMBL6983505 0.79 NR3C1 (0.42) NR3C1ARSLC16A3ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed