SCHEMBL6981070

SCHEMBL6981070

CC1=C(C)C2=C(N)C(C)(CN3CCN(CCc4ccccc4)CC3)CC2=C(C)O1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.41
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
SLC6A3 Q01959 1/20 0.39
HTR1A P08908 1/20 0.39
DRD2 P14416 1/20 0.39
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.38
ACHE P22303 1/20 0.38
OPRM1 P35372 1/20 0.37
KCNH2 Q12809 1/20 0.37
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8578232 0.94 SIGMAR1 (0.46) SIGMAR1MEN1KMT2A
Hydrochloric Acid SCHEMBL6979051 0.88 LMNA (0.41) SIGMAR1MAPTNPSR1DRD2MEN1
SCHEMBL6983492 0.84 CHRNA7 (0.40) SIGMAR1MAPTNPSR1HTR1ADRD2
SCHEMBL6981079 0.84 HRH3 (0.40) SIGMAR1ACHE
Hydrochloric Acid SCHEMBL6982807 0.83 SIGMAR1 (0.42) SIGMAR1SLC6A3HTR1ADRD2MEN1
SCHEMBL6981931 0.83 HRH3 (0.39) SIGMAR1ACHE
SCHEMBL6979708 0.83 PRMT6 (0.43) SIGMAR1KCNH2
Hydrochloric Acid SCHEMBL6985676 0.80 SMN1; SMN2 (0.42) SIGMAR1MAPTNPSR1SLC6A3MEN1
SCHEMBL8573871 0.80 LMNA (0.42) MEN1ALDH1A1KMT2A
Hydrochloric Acid SCHEMBL6984760 0.80 DRD2 (0.40) SIGMAR1HTR1ADRD2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed