SCHEMBL6981732

SCHEMBL6981732

Cc1ccc(NC(=O)CCCN2CCN3CCCCC3C2)cc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
SIGMAR1 Q99720 1/20 0.47
TSHR P16473 1/20 0.47
HTT P42858 1/20 0.47
LMNA P02545 1/20 0.47
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
TP53 P04637 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5842390 0.99 MEN1 (0.56) MEN1KMT2ASIGMAR1TSHRHTT
SCHEMBL5840932 0.89 CACNA1G (0.60) SIGMAR1LMNATP53
SCHEMBL6987296 0.89 ALDH1A1 (0.54) SIGMAR1LMNAALDH1A1
SCHEMBL6986958 0.89 SMN1; SMN2 (0.54) KMT2AHTTLMNATP53ALDH1A1
SCHEMBL6978967 0.89 LMNA (0.53) KMT2ASIGMAR1LMNACYP2C19TP53
SCHEMBL6987557 0.89 HTR1A (0.52) SIGMAR1HRH3CA1CA2CA9
SCHEMBL6980711 0.89 MAPT (0.57) KMT2ATP53HRH3ALDH1A1
Hydrochloric Acid SCHEMBL5842633 0.88 SMN1; SMN2 (0.56) KMT2AHTTLMNATP53ALDH1A1
Hydrochloric Acid SCHEMBL5842876 0.88 KMT2A (0.55) MEN1KMT2ASIGMAR1TSHRLMNA
Hydrochloric Acid SCHEMBL5842086 0.88 HTR1A (0.53) HRH3CA1CA2CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1275647-B1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-11-12 EP disclosed