SCHEMBL6986958

SCHEMBL6986958

O=C(CCCN1CCN2CCCCC2C1)Nc1ccc(Br)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.54
GAA P10253 1/20 0.54
TP53 P04637 3/20 0.51
L3MBTL1 Q9Y468 3/20 0.49
KDM4E B2RXH2 2/20 0.49
HTT P42858 2/20 0.49
LMNA P02545 2/20 0.49
MAPK1 P28482 1/20 0.49
HIF1A Q16665 1/20 0.49
ALDH1A1 P00352 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
HTR7 P34969 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
KMT2A Q03164 1/20 0.47
FPR3 P25089 1/20 0.47
FPR2 P25090 1/20 0.47
CCR2 P41597 1/20 0.46
KCNH2 Q12809 1/20 0.46
CACNA1G O43497 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5842633 0.99 SMN1; SMN2 (0.56) SMN1; SMN2GAATP53L3MBTL1KDM4E
SCHEMBL6987296 0.89 ALDH1A1 (0.54) GAAKDM4ELMNAALDH1A1CACNA1G
SCHEMBL5840932 0.89 CACNA1G (0.60) GAATP53L3MBTL1LMNACACNA1G
SCHEMBL6981732 0.89 MEN1 (0.54) TP53HTTLMNAALDH1A1KMT2A
SCHEMBL6978967 0.89 LMNA (0.53) TP53LMNAALDH1A1KMT2ACACNA1G
Hydrochloric Acid SCHEMBL5842390 0.88 MEN1 (0.56) SMN1; SMN2GAATP53HTTLMNA
Hydrochloric Acid SCHEMBL5842876 0.88 KMT2A (0.55) TP53KDM4ELMNAMAPK1ALDH1A1
SCHEMBL6985625 0.86 CCR2 (0.48) SMN1; SMN2LMNAHTR7FPR3FPR2
SCHEMBL6987557 0.86 HTR1A (0.52) ALDH1A1HTR7CACNA1G
SCHEMBL6980711 0.86 MAPT (0.57) SMN1; SMN2TP53L3MBTL1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1275647-B1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-11-12 EP disclosed
EP-1275647-A1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2003-01-15 EP disclosed