SCHEMBL6980780

SCHEMBL6980780

Cc1c(C)c2c(c(C)c1N)CC(C)(CN1CCN(C(=O)CC(c3ccccc3)c3ccccc3)CC1)O2

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 12/20 0.43
CACNA1B Q00975 12/20 0.43
CACNB1 Q02641 12/20 0.43
CACNA1C Q13936 10/20 0.43
CACNA1H O95180 1/20 0.42
TDP1 Q9NUW8 1/20 0.40
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
CACNA1G O43497 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983244 0.91 CACNA1B (0.35) CACNA2D1CACNA1BCACNB1CACNA1C
SCHEMBL6971808 0.89 HTR7 (0.40) CACNA1CCACNA1G
SCHEMBL6975992 0.88 TSHR (0.44) GAATSHR
SCHEMBL6976114 0.85 USP2 (0.32) TDP1GAATSHR
SCHEMBL6974100 0.83 NPC1 (0.48) CACNA1CTSHR
Hydrochloric Acid SCHEMBL6984860 0.82 OPRL1 (0.37)
SCHEMBL9698183 0.82 OPRM1 (0.38) GAA
Hydrochloric Acid SCHEMBL8713715 0.81 MEN1 (0.38) GAA
Hydrochloric Acid SCHEMBL6982801 0.81 SIGMAR1 (0.41)
SCHEMBL6975786 0.80 POLB (0.40) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed