SCHEMBL6974100

SCHEMBL6974100

Cc1c(C)c2c(c(C)c1N)CC(C)(CN1CCN(C(=O)CCCc3ccccc3)CC1)O2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
SIGMAR1 Q99720 5/20 0.46
AR P10275 1/20 0.45
TSHR P16473 1/20 0.41
CACNA1F O60840 1/20 0.41
DRD1 P21728 1/20 0.41
DRD4 P21917 1/20 0.41
DRD5 P21918 1/20 0.41
HRH2 P25021 1/20 0.41
ADRA1D P25100 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR7 P34969 1/20 0.41
ADRA1A P35348 1/20 0.41
HRH1 P35367 1/20 0.41
ADRA1B P35368 1/20 0.41
OPRM1 P35372 1/20 0.41
DRD3 P35462 1/20 0.41
OPRD1 P41143 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6977655 0.94 TSHR (0.47) NPC1RAB9ASIGMAR1ARTSHR
SCHEMBL6971808 0.88 HTR7 (0.40) NPC1RAB9ASIGMAR1CACNA1FDRD1
SCHEMBL8578227 0.86 SIGMAR1 (0.46) SIGMAR1POLB
Hydrochloric Acid SCHEMBL6984004 0.85 SIGMAR1 (0.45) SIGMAR1ALDH1A1NPSR1POLB
Hydrochloric Acid SCHEMBL6982193 0.84 SIGMAR1 (0.45) SIGMAR1
SCHEMBL6981065 0.83 SIGMAR1 (0.41) SIGMAR1OPRM1SLC6A3ALDH1A1MAPT
SCHEMBL6980780 0.83 CACNA2D1 (0.43) TSHRCACNA1C
SCHEMBL6985365 0.81 LMNA (0.42) NPC1RAB9ASIGMAR1DRD4ALDH1A1
SCHEMBL6981074 0.80 HRH3 (0.40) SIGMAR1OPRK1
SCHEMBL6981926 0.80 HRH3 (0.39) SIGMAR1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed