SCHEMBL6982220

SCHEMBL6982220

O=S(=O)(Nc1cccc2c1NCCC2)c1ccc(Cl)cc1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.64
LMNA P02545 2/20 0.64
KDM4E B2RXH2 1/20 0.64
GAA P10253 1/20 0.64
HTT P42858 1/20 0.64
SLC40A1 Q9NP59 1/20 0.48
CYP19A1 P11511 1/20 0.44
BRD4 O60885 1/20 0.43
HTR2C P28335 2/20 0.43
HTR2B P41595 1/20 0.43
CCR2 P41597 1/20 0.42
CES1 P23141 1/20 0.42
HKDC1 Q2TB90 1/20 0.41
DRD2 P14416 1/20 0.41
HTR2A P28223 1/20 0.41
DRD3 P35462 1/20 0.41
HTR6 P50406 1/20 0.41
KCNA5 P22460 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6984823 0.88 HTR6 (0.48) ALDH1A1LMNAKDM4EGAAHTT
SCHEMBL6983864 0.88 SLC40A1 (0.50) ALDH1A1LMNAKDM4EGAAHTT
SCHEMBL6985112 0.87 ALDH1A1 (0.64) ALDH1A1LMNAKDM4EGAAHTT
SCHEMBL6986762 0.87 ALDH1A1 (0.53) ALDH1A1LMNAKDM4EGAAHTT
SCHEMBL6985321 0.87 ALDH1A1 (0.48) ALDH1A1LMNAKDM4EGAAHTT
SCHEMBL6976544 0.81 MEN1 (0.53) ALDH1A1LMNAHTTHTR2CHTR2B
SCHEMBL6974140 0.80 WDR5 (0.45) ALDH1A1LMNAKDM4EGAAHTT
SCHEMBL30926919 0.75 ALDH1A1 (0.55) ALDH1A1LMNAKDM4EGAAHTT
SCHEMBL27181380 0.75 ALDH1A1 (0.55) ALDH1A1LMNAKDM4EGAAHTT
SCHEMBL6983098 0.75 HCRTR1 (0.43) ALDH1A1LMNAGAAHTR6KCNA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed