SCHEMBL6982483

SCHEMBL6982483

O=C(O)C1(c2ccc(Cl)cc2)OCC2(CO1)c1ccccc1C=Cc1ccccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 4/20 0.44
HSD11B1 P28845 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
HIF1A Q16665 1/20 0.35
CCR1 P32246 1/20 0.34
LMNA P02545 3/20 0.34
ALDH1A1 P00352 2/20 0.33
HTT P42858 2/20 0.33
SCN9A Q15858 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CNR1 P21554 1/20 0.33
MAPK1 P28482 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
HSD17B3 P37058 1/20 0.32
HDAC4 P56524 1/20 0.32
CES2 O00748 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6971210 0.86 CYP1A2 (0.41) KIF11HSD11B1SMN1; SMN2TP53CYP1A2
SCHEMBL6974413 0.84 HRH1 (0.37) KIF11SMN1; SMN2TP53CYP1A2CYP2C19
SCHEMBL6967893 0.83 CNR1 (0.40) HSD11B1ALDH1A1CNR1MAPK1CES2
SCHEMBL6970254 0.82 OPRM1 (0.41) KIF11HSD11B1SMN1; SMN2LMNAALDH1A1
SCHEMBL377756 0.81 MAPK1 (0.40) HSD11B1ALDH1A1CNR1MAPK1HDAC4
SCHEMBL6982681 0.76 THRB (0.44) KIF11ALDH1A1NPSR1HDAC4
SCHEMBL6975695 0.75 POLB (0.38) HSD11B1CYP1A2CYP2C19ALDH1A1HTT
SCHEMBL6976918 0.75 HSD11B1 (0.40) HSD11B1LMNAALDH1A1MAPK1HDAC4
SCHEMBL7145811 0.73 APP (0.38) SMN1; SMN2LMNAALDH1A1HTTMAPK1
SCHEMBL6981777 0.73 AKR1C1 (0.41) SMN1; SMN2LMNAALDH1A1HTTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1098893-B1 CYCLIC COMPOUNDS USEFUL IN THE TREATMENT OF DYSLIPIDEMIA, ATHEROSCLEROSIS AND DIABETES, PHARMACEUTICAL COMPOSITIONS AND PREPARATION PROCESS MERCK PATENT GMBH (DE) 2003-03-26 EP disclosed
US-6528538-B1 Reaction of 1,3-propanediol derivative with a ketone or aldehyde MERCK PATENTGESELLSCHAFT (DE) 2003-03-04 US disclosed