SCHEMBL6983189

SCHEMBL6983189

Fc1ccc([C](CCc2ccccc2)Cc2cccc(Cl)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 3/20 0.50
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
CTSL P07711 2/20 0.44
CTSB P07858 2/20 0.44
PLAAT3 P53816 2/20 0.44
PLAAT5 Q96KN8 2/20 0.44
PLAAT2 Q9NWW9 2/20 0.44
PLAAT4 Q9UL19 2/20 0.44
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 1/20 0.44
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
HTR3A P46098 1/20 0.42
HTR3D Q70Z44 1/20 0.42
HTR3C Q8WXA8 1/20 0.42
CTBP2 P56545 1/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983635 0.85 ALDH1A1 (0.53) PLAAT3PLAAT5PLAAT2PLAAT4ALDH1A1
SCHEMBL6985463 0.79 L3MBTL1 (0.56) GRIN2BPLAAT3PLAAT5PLAAT2PLAAT4
SCHEMBL6979677 0.75 CTSL (0.52) CTSLCTSBALDH1A1KDM4EMEN1
SCHEMBL8956360 0.75 GRIN2B (0.56) GRIN2BCYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL13561129 0.73 PLAAT3 (0.57) CTSLCTSBPLAAT3PLAAT5PLAAT2
SCHEMBL8329374 0.71 CTSL (0.51) GRIN2BCTSLCTSBPLAAT3PLAAT5
SCHEMBL11697150 0.70 F2 (0.51) GRIN2BCYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL23071686 0.69 TAAR1 (0.65) CYP3A4PLAAT3PLAAT5PLAAT2PLAAT4
SCHEMBL6985694 0.69 ALDH1A1 (0.55) PLAAT3PLAAT5PLAAT2PLAAT4ALDH1A1
SCHEMBL28012695 0.67 NPC1 (0.65) PLAAT3PLAAT5PLAAT2PLAAT4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294695-A2 SUBSTITUTED DIAMIDE DERIVATIVES USEFUL AS MOTILIN ANTAGONISTS Ortho-McNeil Pharmaceutical, Inc. (US) 2003-03-26 EP disclosed
WO-2001085694-A2 SUBSTITUTED DIAMIDE DERIVATIVES USEFUL AS MOTILIN ANTAGONISTS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-11-15 WO disclosed