SCHEMBL6983492

SCHEMBL6983492

CC1=C(C)C2=C(N)C(C)(CN3CCN(c4ccccc4)CC3)CC2=C(C)O1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.40
DRD2 P14416 2/20 0.38
SIGMAR1 Q99720 1/20 0.38
CYP2D6 P10635 1/20 0.36
KCNH2 Q12809 2/20 0.36
DRD4 P21917 2/20 0.36
HTR7 P34969 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
GFER P55789 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HTR1A P08908 1/20 0.35
DRD3 P35462 1/20 0.34
EGFR P00533 1/20 0.34
LMNA P02545 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6979051 0.85 LMNA (0.41) DRD2SIGMAR1DRD4ALDH1A1MAPT
SCHEMBL8578232 0.83 SIGMAR1 (0.46) SIGMAR1
Hydrochloric Acid SCHEMBL6980233 0.82 CHRNA7 (0.39) CHRNA7DRD2SIGMAR1KCNH2DRD4
Hydrochloric Acid SCHEMBL6984760 0.81 DRD2 (0.40) DRD2SIGMAR1CYP2D6HTR7HTR1A
Hydrochloric Acid SCHEMBL6985853 0.81 DRD2 (0.40) DRD2SIGMAR1CYP2D6HTR7HTR1A
SCHEMBL6979708 0.81 PRMT6 (0.43) SIGMAR1KCNH2
SCHEMBL8573871 0.80 LMNA (0.42) ALDH1A1KDM4EL3MBTL1LMNA
Hydrochloric Acid SCHEMBL6981605 0.78 MEN1 (0.41) DRD2CYP2D6KCNH2ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL6985676 0.78 SMN1; SMN2 (0.42) SIGMAR1CYP2D6ALDH1A1MAPTLMNA
Hydrochloric Acid SCHEMBL6981674 0.78 SIGMAR1 (0.38) DRD2SIGMAR1DRD4ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed