SCHEMBL6984595

SCHEMBL6984595

CC(C)C[C@@H](C(=O)NN(CCCCNC(=O)OCc1ccccc1)Cc1ccccc1)[C@H](CCCc1ccccc1)C(=O)NOC1CCCCO1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.37
MMP3 P08254 1/20 0.37
CTSL P07711 2/20 0.36
CTSS P25774 2/20 0.36
CTSK P43235 2/20 0.36
CPB1 P15086 1/20 0.36
CPB2 Q96IY4 1/20 0.36
DPP8 Q6V1X1 2/20 0.35
DPP7 Q9UHL4 2/20 0.35
DPP4 P27487 1/20 0.35
DPP9 Q86TI2 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35
ANPEP P15144 1/20 0.35
KLK7 P49862 2/20 0.35
KLK5 Q9Y337 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6986871 0.89 MMP1 (0.37) MMP3
SCHEMBL6982715 0.89 CYP1A2 (0.37) CYP1A2MMP3CTSLCTSSCTSK
SCHEMBL6986124 0.82 CTSS (0.36) CYP1A2CTSLCTSSCTSK
SCHEMBL6940058 0.82 CTSK (0.38) CYP1A2MMP3CTSLCTSSCTSK
SCHEMBL7840445 0.79 MMP1 (0.46) MMP3
SCHEMBL6942326 0.79 MMP1 (0.39) MMP3
SCHEMBL6983815 0.78 MMP1 (0.41) CYP1A2MMP3
SCHEMBL6982858 0.76 MMP1 (0.38) CTSL
SCHEMBL6984591 0.75 CTSK (0.38) CYP1A2MMP3CTSLCTSSCTSK
SCHEMBL6982289 0.75 MMP1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1089964-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-10-29 EP disclosed
US-6239151-B1 TREATMENT OF INFLAMMATORY AND AUTOIMMUNE DISEASES, OSTEOARTHRITIS, RESPIRATORY DISEASES, TUMORS, CACHEXIA, CARDIOVASCULAR DISEASES, FEVER, HAEMORRHAGE AND SEPSIS, HYDRAZINE DERIVATIVES, HOFFMANN-LA ROCHE INC. 2001-05-29 US disclosed