SCHEMBL6985214

SCHEMBL6985214

CCCc1c[nH]c2ccc(Oc3c(C)cc(O)cc3Br)cc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.45
HTR1A P08908 9/20 0.45
HTR1B P28222 8/20 0.45
HTR2A P28223 3/20 0.45
HTR1D P28221 8/20 0.43
TRPM8 Q7Z2W7 2/20 0.43
CYP1A2 P05177 2/20 0.43
MAPT P10636 2/20 0.43
MTNR1A P48039 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43
HTR2C P28335 1/20 0.43
HTR7 P34969 1/20 0.43
HTR6 P50406 1/20 0.43
HTR4 Q13639 1/20 0.43
KDM4E B2RXH2 1/20 0.42
TP53 P04637 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6987620 0.85 THRA (0.45) CYP2D6HTR1AHTR1BHTR2AHTR1D
SCHEMBL7089914 0.84 THRA (0.47) CYP2D6HTR1AHTR1BHTR2AHTR1D
SCHEMBL6523679 0.83 KDM4E (0.49) HTR1AHTR1BHTR1DTRPM8MTNR1A
SCHEMBL6513222 0.83 KDM4E (0.46) CYP2D6HTR1AHTR1BHTR2AHTR1D
SCHEMBL7090401 0.82 HTR1A (0.52) CYP2D6HTR1AHTR1BHTR2AHTR1D
SCHEMBL7089278 0.80 HTR1A (0.52) CYP2D6HTR1AHTR1BHTR2AHTR1D
SCHEMBL6983004 0.79 HTR1A (0.45) CYP2D6HTR1AHTR1BHTR2AHTR1D
SCHEMBL6862010 0.78 KDM4E (0.53) HTR1AHTR1BHTR1DMTNR1AKDM4E
SCHEMBL6989252 0.78 HTR2B (0.49) CYP2D6HTR1AHTR1BHTR2AHTR1D
SCHEMBL6985820 0.78 THRA (0.46) CYP2D6HTR1AHTR1BHTR2AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347959-A1 INDOLE DERIVATIVES AS LIGANDS OF THYROID RECEPTORS Bayer Aktiengesellschaft (DE) 2003-10-01 EP disclosed
WO-2002051805-A1 INDOLE DERIVATIVES AS LIGANDS OF THYROID RECEPTORS BAYER AKTIENGESELLSCHAFT (DE) 2002-07-04 WO disclosed