SCHEMBL6985422

SCHEMBL6985422

COc1ccc(NC(=O)CCCN2CCN3CCCCC3C2)cc1OC

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SHMT2 P34897 1/20 0.64
NPSR1 Q6W5P4 2/20 0.55
ALDH1A1 P00352 4/20 0.51
LMNA P02545 4/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
MAPT P10636 2/20 0.48
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
POLB P06746 1/20 0.46
ATM Q13315 1/20 0.46
CACNA1G O43497 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5840743 0.99 SHMT2 (0.63) SHMT2NPSR1ALDH1A1LMNASMN1; SMN2
SCHEMBL6986043 0.89 SHMT2 (0.50) SHMT2NPSR1ALDH1A1LMNASMN1; SMN2
Hydrochloric Acid SCHEMBL5843596 0.89 SHMT2 (0.49) SHMT2ALDH1A1LMNASMN1; SMN2MAPT
SCHEMBL6980711 0.87 MAPT (0.57) ALDH1A1SMN1; SMN2MAPTKMT2AL3MBTL1
Hydrochloric Acid SCHEMBL5842053 0.86 MAPT (0.56) ALDH1A1SMN1; SMN2MAPTKMT2AL3MBTL1
SCHEMBL6981732 0.84 MEN1 (0.54) ALDH1A1LMNAMEN1KMT2A
SCHEMBL6985937 0.83 NPSR1 (0.59) NPSR1ALDH1A1LMNASMN1; SMN2MAPT
SCHEMBL6985243 0.83 SHMT2 (0.52) SHMT2NPSR1ALDH1A1LMNAMAPT
SCHEMBL5842521 0.83 SIGMAR1 (0.57) L3MBTL1CACNA1G
Hydrochloric Acid SCHEMBL5842390 0.83 MEN1 (0.56) ALDH1A1LMNASMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1275647-B1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-11-12 EP disclosed
EP-1275647-A1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2003-01-15 EP disclosed