SCHEMBL6985937

SCHEMBL6985937

COc1ccccc1NC(=O)CCCN1CCN2CCCCC2C1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.59
L3MBTL1 Q9Y468 2/20 0.56
ALDH1A1 P00352 2/20 0.53
HTR1A P08908 4/20 0.52
HTR7 P34969 4/20 0.52
THRB P10828 1/20 0.51
TSHR P16473 2/20 0.50
USP2 O75604 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
HTT P42858 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
MEN1 O00255 1/20 0.49
LMNA P02545 1/20 0.49
MAPT P10636 1/20 0.49
KMT2A Q03164 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5842200 0.99 NPSR1 (0.58) NPSR1L3MBTL1ALDH1A1HTR1AHTR7
SCHEMBL6985422 0.83 SHMT2 (0.64) NPSR1L3MBTL1ALDH1A1SMN1; SMN2MEN1
Hydrochloric Acid SCHEMBL5840743 0.83 SHMT2 (0.63) NPSR1L3MBTL1ALDH1A1HTR1AHTR7
SCHEMBL6986827 0.83 SIGMAR1 (0.47)
SCHEMBL6986043 0.82 SHMT2 (0.50) NPSR1L3MBTL1ALDH1A1THRBSMN1; SMN2
SCHEMBL6978967 0.82 LMNA (0.53) ALDH1A1CYP2C19LMNAKMT2A
SCHEMBL6980711 0.82 MAPT (0.57) L3MBTL1ALDH1A1SMN1; SMN2MAPTKMT2A
Hydrochloric Acid SCHEMBL5842696 0.82 CHRM2 (0.49)
Hydrochloric Acid SCHEMBL5843596 0.82 SHMT2 (0.49) L3MBTL1ALDH1A1HTR1AHTR7THRB
Hydrochloric Acid SCHEMBL5842876 0.81 KMT2A (0.55) ALDH1A1TSHRMEN1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1275647-B1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-11-12 EP disclosed
EP-1275647-A1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2003-01-15 EP disclosed