SCHEMBL6985790

SCHEMBL6985790

N=C(N)c1ccc(OCC(=O)N2CCCc3cccc(N(CC(=O)O)S(=O)(=O)c4cccc5ccccc45)c32)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 4/20 0.46
NFE2L2 Q16236 4/20 0.46
F2 P00734 5/20 0.41
ITGB3 P05106 3/20 0.38
ITGA2B P08514 3/20 0.38
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36
MAPT P10636 3/20 0.35
TP53 P04637 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
TSHR P16473 1/20 0.35
TPSAB1 Q15661 1/20 0.35
TPSD1 Q9BZJ3 1/20 0.35
TPSG1 Q9NRR2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6978680 0.87 KEAP1 (0.47) KEAP1NFE2L2F2ITGB3ITGA2B
SCHEMBL6982918 0.86 F2 (0.47) KEAP1NFE2L2F2MEN1ALDH1A1
SCHEMBL7084264 0.79 F2 (0.40) KEAP1NFE2L2F2ITGB3ITGA2B
SCHEMBL6979635 0.76 ITGB3 (0.40) KEAP1NFE2L2F2ITGB3ITGA2B
SCHEMBL6978671 0.73 F2 (0.46) KEAP1NFE2L2F2ITGB3ITGA2B
SCHEMBL6976368 0.72 ITGB3 (0.39) F2ITGB3ITGA2BTPSAB1TPSD1
SCHEMBL6982923 0.72 ALDH1A1 (0.40) MEN1ALDH1A1KMT2AMAPTTP53
SCHEMBL6984709 0.72 F2 (0.44) KEAP1NFE2L2F2ITGB3ITGA2B
Hydrochloric Acid SCHEMBL6982383 0.72 ALDH1A1 (0.39) F2MEN1ALDH1A1KMT2AMAPT
SCHEMBL6985025 0.71 F7 (0.42) F2ITGB3ITGA2BTPSAB1TPSD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP claimed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP claimed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO claimed
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed