SCHEMBL6978680

SCHEMBL6978680

N=C(N)c1ccc(CCC(=O)N2CCCc3cccc(N(CC(=O)O)S(=O)(=O)c4cccc5ccccc45)c32)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 4/20 0.47
NFE2L2 Q16236 4/20 0.47
F2 P00734 6/20 0.40
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
F10 P00742 2/20 0.35
SLC16A3 O15427 1/20 0.35
PLG P00747 1/20 0.35
PRSS1 P07477 1/20 0.35
TPSAB1 Q15661 1/20 0.35
TPSD1 Q9BZJ3 1/20 0.35
TPSG1 Q9NRR2 1/20 0.35
PTGER4 P35408 1/20 0.34
PTGER2 P43116 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7084264 0.92 F2 (0.40) KEAP1NFE2L2F2ITGB3ITGA2B
SCHEMBL6979635 0.90 ITGB3 (0.40) KEAP1NFE2L2F2ITGB3ITGA2B
SCHEMBL6985790 0.87 KEAP1 (0.46) KEAP1NFE2L2F2ITGB3ITGA2B
SCHEMBL6976368 0.86 ITGB3 (0.39) F2ITGB3ITGA2BF10PLG
SCHEMBL6978671 0.86 F2 (0.46) KEAP1NFE2L2F2ITGB3ITGA2B
SCHEMBL6985025 0.84 F7 (0.42) F2ITGB3ITGA2BF10PLG
SCHEMBL6984709 0.83 F2 (0.44) KEAP1NFE2L2F2ITGB3ITGA2B
SCHEMBL6981750 0.82 AVPR2 (0.38) KEAP1NFE2L2F2ITGB3ITGA2B
SCHEMBL6982999 0.81 ALDH1A1 (0.41) F2ITGB3ITGA2BPLGPRSS1
SCHEMBL6982234 0.80 TP53 (0.41) F2F10PLGPRSS1TPSAB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP claimed
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed