SCHEMBL6985836

SCHEMBL6985836

CCNc1c(C)c(C)c2c(c1C)CC(C)(CN1CCN(c3ccccc3)CC1)O2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.40
SIGMAR1 Q99720 1/20 0.40
CHRNA7 P36544 1/20 0.39
USP2 O75604 1/20 0.35
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
NFKB1 P19838 1/20 0.35
THPO P40225 1/20 0.35
HIF1A Q16665 1/20 0.35
LCK P06239 1/20 0.35
FYN P06241 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADRA1D P25100 1/20 0.35
MAPK3 P27361 1/20 0.35
HTR2C P28335 1/20 0.35
MC4R P32245 1/20 0.35
HRH1 P35367 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6980227 0.99 DRD2 (0.40) DRD2SIGMAR1CHRNA7USP2TP53
SCHEMBL6983850 0.85 MEN1 (0.39) DRD2USP2HTR2CDRD3HTR2B
Hydrochloric Acid SCHEMBL6980238 0.84 ALDH1A1 (0.40) DRD2USP2HTR2CDRD3HTR2B
SCHEMBL6982079 0.84 DRD2 (0.43) DRD2SIGMAR1DRD3KMT2AHTR7
SCHEMBL6983488 0.83 DRD2 (0.41) DRD2SIGMAR1CHRNA7USP2TP53
SCHEMBL4035933 0.83 ALOX15 (0.50) DRD2SIGMAR1CHRNA7USP2TP53
Hydrochloric Acid SCHEMBL6979630 0.79 SMN1; SMN2 (0.39) SIGMAR1TP53CYP2C9ALOX15TSHR
SCHEMBL2911210 0.78 DRD4 (0.37) DRD2SIGMAR1CHRNA7USP2TP53
SCHEMBL8309041 0.75 HTR2A (0.41) DRD2SIGMAR1TSHRHTR2CDRD3
SCHEMBL9689567 0.72 CYP3A4 (0.63) DRD2USP2TP53CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed