SCHEMBL6986827

SCHEMBL6986827

COc1ccccc1NCCCCN1CCN2CCCCC2C1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.47
CHRM2 P08172 2/20 0.47
CHRM4 P08173 1/20 0.45
ABCB1 P08183 1/20 0.45
CHRM5 P08912 1/20 0.45
ADRA2A P08913 1/20 0.45
CHRM1 P11229 1/20 0.45
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
CHRM3 P20309 1/20 0.45
KCNH2 Q12809 1/20 0.45
TMEM97 Q5BJF2 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5842696 0.99 CHRM2 (0.49) SIGMAR1CHRM2CHRM4ABCB1CHRM5
SCHEMBL5841796 0.84 SIGMAR1 (0.51) SIGMAR1ABCB1TMEM97
Hydrochloric Acid SCHEMBL5840933 0.83 SIGMAR1 (0.50) SIGMAR1ABCB1TMEM97
SCHEMBL6982261 0.83 SHMT2 (0.55) SIGMAR1
SCHEMBL7936484 0.83 SIGMAR1 (0.55) SIGMAR1CHRM2CHRM4ABCB1CHRM5
SCHEMBL6985937 0.83 NPSR1 (0.59)
Hydrochloric Acid SCHEMBL5841553 0.82 SHMT2 (0.54) SIGMAR1
Hydrochloric Acid SCHEMBL5842200 0.82 NPSR1 (0.58)
SCHEMBL5841208 0.82 SHMT2 (0.44) SIGMAR1CHRM2CHRM4ABCB1CHRM5
SCHEMBL6987164 0.82 SIGMAR1 (0.46) SIGMAR1ABCB1TMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1275647-B1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-11-12 EP disclosed
EP-1275647-A1 Octahydro-2H-pyrido[1,2-a]pyrazine derivatives, process for their preparation and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2003-01-15 EP disclosed