SCHEMBL7936484

SCHEMBL7936484

COc1ccccc1NCCN1CCN(C2CCCCC2)CC1

nearest known ligand 0.79

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.55
ABCB1 P08183 2/20 0.51
CHRM2 P08172 1/20 0.51
CHRM4 P08173 1/20 0.51
CHRM5 P08912 1/20 0.51
ADRA2A P08913 1/20 0.51
CHRM1 P11229 1/20 0.51
ADRA2B P18089 1/20 0.51
ADRA2C P18825 1/20 0.51
CHRM3 P20309 1/20 0.51
KCNH2 Q12809 1/20 0.51
TMEM97 Q5BJF2 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6986827 0.83 SIGMAR1 (0.47) SIGMAR1ABCB1CHRM2CHRM4CHRM5
SCHEMBL4930910 0.83 ACHE (0.62) CHRM2
Hydrochloric Acid SCHEMBL5842696 0.82 CHRM2 (0.49) SIGMAR1ABCB1CHRM2CHRM4CHRM5
SCHEMBL23338779 0.78 SIGMAR1 (0.51) SIGMAR1ABCB1TMEM97
SCHEMBL6930794 0.77 DRD2 (0.66)
SCHEMBL23339263 0.71 SIGMAR1 (0.52) SIGMAR1ABCB1CHRM2CHRM4CHRM5
SCHEMBL29985090 0.71 SIGMAR1 (1.00) SIGMAR1ABCB1CHRM2CHRM4CHRM5
SCHEMBL8711292 0.71 CYP2D6 (0.71)
SCHEMBL4072190 0.70 L3MBTL1 (0.51) SIGMAR1KCNH2
SCHEMBL4923558 0.70 ALDH1A1 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235732-B1 RESPIRATORY SYSTEM DISORDERS; ANTIINFLAMMATORY AGENTS; SKIN DISORDERS BOEHRINGER INGELHEIM KG (DE) 2001-05-22 US disclosed
US-6191135-B1 Neurokinin antagonists BOEHRINGER INGELHEIM KG (DE) 2001-02-20 US disclosed
US-5985881-A TREATMENT AND PREVENTION OF RESPIRATORY DISORDERS, INFLAMMATORY EYE DISEASES, INFLAMMATORY SKIN DISEASES, INTESTINAL DISORDERS, OTHER INFLAMMATORY DISEASES BOEHRINGER INGELHEIM KG (DE) 1999-11-16 US disclosed
US-5708006-A ANTIINFLAMMATORY AGENTS BOEHRINGER INGELHEIM KG (DE) 1998-01-13 US disclosed
US-5696123-A ALPHA-PIPERAZINYL BENZYL COMPOUND AS TACHYKININ ANTAGONIST TREATING ASTHMA, BRONCHITIS, SKIN DISORDER, EYE DISEASE, HEADACHE, GASTROINTESTINAL DISORDER BOEHRINGER INGELHEIM KG (DE) 1997-12-09 US disclosed