SCHEMBL6987482

SCHEMBL6987482

CC(C)N1CCC(CCNC(=O)CNc2cccc(C(=O)c3ccc4cc[nH]c4c3)c2Cl)CC1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.37
F10 P00742 2/20 0.36
MAPK11 Q15759 1/20 0.35
MAPK14 Q16539 1/20 0.35
HRH3 Q9Y5N1 2/20 0.35
HTR4 Q13639 3/20 0.34
ACHE P22303 2/20 0.34
SIGMAR1 Q99720 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
ALOX12 P18054 1/20 0.34
HSD17B10 Q99714 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
NR4A2 P43354 1/20 0.34
VCP P55072 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985512 0.80 KDM4E (0.45) SMYD3F10KDM4EALDH1A1MAPT
SCHEMBL6989019 0.75 FAAH (0.42) F10HRH3HTR4ACHEALDH1A1
SCHEMBL5868417 0.74 SMYD3 (0.38) SMYD3F10MAPK14HRH3HTR4
Hydrochloric Acid SCHEMBL5868316 0.73 F10 (0.36) SMYD3F10MAPK11MAPK14HRH3
SCHEMBL6987333 0.73 PYGL (0.42) SMYD3HRH3HTR4VCP
SCHEMBL6986945 0.72 F10 (0.53) SMYD3F10MAPK14KDM4EALDH1A1
Hydrochloric Acid SCHEMBL6985167 0.72 F10 (0.53) SMYD3F10MAPK14HRH3KDM4E
SCHEMBL6988752 0.70 ALDH1A1 (0.43) SMYD3F10HTR4SIGMAR1KDM4E
Trifluoroacetic Acid SCHEMBL5868462 0.70 F10 (0.36) SMYD3F10MAPK11MAPK14HRH3
SCHEMBL5868347 0.70 SMYD3 (0.35) SMYD3F10HRH3HTR4ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289954-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2003-03-12 EP disclosed
WO-2001096303-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2001-12-20 WO disclosed