SCHEMBL6987333

SCHEMBL6987333

CC(C)N1CCC(CNC(=O)CNc2cccc(C(=O)c3cc4cc(Cl)ccc4[nH]3)c2Cl)CC1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PYGL P06737 14/20 0.42
VCP P55072 1/20 0.40
SMYD3 Q9H7B4 2/20 0.40
HRH4 Q9H3N8 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
HTR4 Q13639 1/20 0.39
NHERF1 O14745 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6990232 0.88 PYGL (0.42) PYGLSMYD3HRH4NHERF1
SCHEMBL6984406 0.87 CHRM1 (0.44) PYGLSMYD3HRH4NHERF1
SCHEMBL6989019 0.77 FAAH (0.42) HRH3HTR4
SCHEMBL5868411 0.74 PYGL (0.43) PYGLSMYD3HRH4HRH3
SCHEMBL6987482 0.73 SMYD3 (0.37) VCPSMYD3HRH3HTR4
Trifluoroacetic Acid SCHEMBL5867893 0.72 PYGL (0.44) PYGLSMYD3
SCHEMBL6984041 0.69 ROCK2 (0.43) HRH3HTR4
SCHEMBL6987182 0.68 FAAH (0.43) HRH3HTR4
SCHEMBL6985512 0.68 KDM4E (0.45) SMYD3
Hydrochloric Acid SCHEMBL6984317 0.67 ROCK2 (0.44) HRH3HTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289954-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2003-03-12 EP disclosed
WO-2001096303-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2001-12-20 WO disclosed