SCHEMBL6988714

SCHEMBL6988714

CC(C)(CNC(=O)c1cccc(-c2cccnc2)c1)CNc1c(Nc2cccnc2)c(=O)c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.43
CDK4 P11802 1/20 0.42
CCND1 P24385 1/20 0.42
KMO O15229 1/20 0.42
EGFR P00533 2/20 0.42
TBXA2R P21731 1/20 0.42
TBXAS1 P24557 1/20 0.42
MEN1 O00255 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
ABL1 P00519 2/20 0.41
SRC P12931 1/20 0.41
ROCK2 O75116 2/20 0.40
BCR P11274 1/20 0.40
BLK P51451 1/20 0.39
BTK Q06187 1/20 0.39
SMPD1 P17405 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PSMD14 O00487 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6986333 0.89 MEN1 (0.48) TBXA2RTBXAS1MEN1RAB9AKMT2A
SCHEMBL6987131 0.89 GRM5 (0.44) TBXA2RTBXAS1MEN1KMT2AALDH1A1
SCHEMBL6988050 0.88 ALPL (0.43) TBXA2RTBXAS1MEN1RAB9AKMT2A
SCHEMBL6990458 0.85 CSF1R (0.44) TBXA2RTBXAS1MEN1RAB9AKMT2A
SCHEMBL6988688 0.85 ABCC9 (0.41) TBXA2RTBXAS1RAB9AL3MBTL1MAPKAPK2
SCHEMBL6988180 0.84 NAMPT (0.51) RAB9AKMT2AALDH1A1POLB
SCHEMBL6981925 0.83 NAMPT (0.50) MEN1RAB9AKMT2A
SCHEMBL6989487 0.83 ALDH1A1 (0.49) MEN1RAB9AKMT2AALDH1A1POLB
SCHEMBL4367794 0.79 GRM5 (0.45) MEN1RAB9AKMT2A
SCHEMBL6988709 0.78 CYP1A2 (0.46) SIRT2KMOEGFRTBXA2RTBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358160-A1 AMINAL DIONES AS POTASSIUM CHANNEL OPENERS Abbott Laboratories (US) 2003-11-05 EP disclosed
WO-2002062761-A1 AMINAL DIONES AS POTASSIUM CHANNEL OPENERS ABBOTT LABORATORIES (US) 2002-08-15 WO disclosed