SCHEMBL6990649

SCHEMBL6990649

CCCC(C)(C)Oc1ccc(C(=O)N2CCCCc3sccc32)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 10/20 0.50
AVPR1B P47901 8/20 0.50
AVPR2 P30518 7/20 0.46
ALDH1A1 P00352 5/20 0.43
HPGD P15428 4/20 0.43
TSHR P16473 3/20 0.43
MAPT P10636 2/20 0.43
POLB P06746 1/20 0.43
OXTR P30559 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.40
MITF O75030 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
THRB P10828 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7093443 0.84 ALDH1A1 (0.58) AVPR1AAVPR1BAVPR2ALDH1A1HPGD
SCHEMBL6991852 0.78 AVPR1A (0.49) AVPR1AAVPR1BAVPR2ALDH1A1HPGD
SCHEMBL6991585 0.77 AVPR1A (0.50) AVPR1AAVPR1BAVPR2ALDH1A1HPGD
SCHEMBL6991806 0.76 AVPR1A (0.47) AVPR1AAVPR1BAVPR2ALDH1A1HPGD
SCHEMBL6985203 0.75 AVPR1A (0.61) AVPR1AAVPR1BAVPR2OXTR
SCHEMBL6988048 0.75 NAAA (0.55) AVPR1AAVPR1BAVPR2ALDH1A1HPGD
SCHEMBL6989910 0.75 AVPR1A (0.46) AVPR1AAVPR1BAVPR2ALDH1A1HPGD
SCHEMBL4146200 0.73 AVPR1A (0.68) AVPR1AAVPR1BAVPR2HPGDOXTR
SCHEMBL7365160 0.72 AVPR1A (0.68) AVPR1AAVPR1BAVPR2MAPTPOLB
SCHEMBL6987431 0.72 AVPR1A (0.60) AVPR1AAVPR1BAVPR2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0811008-B1 BICYCLIC BENZAZEPINE DERIVATIVES AS VASOPRESSIN ANTAGONISTS WYETH CORP (US) 2003-10-01 EP disclosed