SCHEMBL6992361

SCHEMBL6992361

CC1CN(c2ccc(-c3nc4cc(Cl)ccc4[nH]3)cn2)CCN1c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 16/20 0.46
KCNH2 Q12809 9/20 0.46
ADORA2A P29274 3/20 0.46
CYP2C9 P11712 1/20 0.42
TRPV1 Q8NER1 1/20 0.42
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40
DHFR P00374 1/20 0.40
NPC1 O15118 1/20 0.40
SOAT1 P35610 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6994712 0.85 DGAT1 (0.54) DGAT1KCNH2ADORA2ACYP2C9DRD2
SCHEMBL6993769 0.76 CHEK2 (0.53) DGAT1KCNH2ADORA2ACYP2C9DRD2
SCHEMBL1687841 0.76 HTR3E (0.54) DGAT1KCNH2ADORA2ACYP2C9NPC1
SCHEMBL14128550 0.76 DGAT1 (0.59) DGAT1KCNH2ADORA2ACYP2C9NPC1
SCHEMBL4560992 0.75 DGAT1 (0.57) DGAT1KCNH2ADORA2ACYP2C9SOAT1
SCHEMBL4566255 0.74 DGAT1 (0.49) DGAT1KCNH2ADORA2ACYP2C9NPC1
SCHEMBL6994359 0.74 CHEK2 (0.50) DGAT1KCNH2ADORA2ACYP2C9DRD2
SCHEMBL10081917 0.74 DGAT1 (0.51) DGAT1KCNH2ADORA2ACYP2C9SOAT1
SCHEMBL4562113 0.74 DGAT1 (0.52) DGAT1KCNH2ADORA2ACYP2C9DRD2
SCHEMBL4543095 0.73 DGAT1 (0.53) DGAT1KCNH2ADORA2ACYP2C9SOAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064569-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-05-18 WO disclosed