SCHEMBL7001083

SCHEMBL7001083

O=C(c1ccc(Cl)cc1)C1CNCCC1(O)CCc1ccc(Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
MBTPS1 Q14703 1/20 0.39
DRD2 P14416 1/20 0.36
KCNH2 Q12809 2/20 0.36
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6995095 0.83 SLC6A3 (0.45) KCNH2
SCHEMBL6998084 0.76 HTR2A (0.38) ALDH1A1LMNAMAPTKMT2A
SCHEMBL7001284 0.73 LMNA (0.44) ALDH1A1LMNAMAPTKMT2ADRD2
SCHEMBL7001738 0.65 ALDH1A1 (0.36) ALDH1A1LMNAMAPTKMT2APOLB
SCHEMBL4239004 0.64 RARB (0.41) ALDH1A1MAPTKMT2A
SCHEMBL6841616 0.63 LMNA (0.53) ALDH1A1LMNAMAPTKMT2AKDM4E
SCHEMBL7769506 0.63 MEN1 (0.43) ALDH1A1LMNAMAPTKMT2AKDM4E
SCHEMBL4674968 0.63 DRD2 (0.53) ALDH1A1LMNAMAPTKMT2ADRD2
SCHEMBL4671412 0.62 MGLL (0.49) LMNAMAPTKMT2AKDM4E
SCHEMBL8967555 0.62 KMT2A (0.56) ALDH1A1LMNAMAPTKMT2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP claimed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP claimed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO claimed
EP-1242080-A4 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE UNIV GEORGETOWN (US) 2003-01-22 EP disclosed
EP-1242080-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2002-09-25 EP disclosed
WO-2001022964-A1 DOPAMINE TRANSPORTER INHIBITORS AND THEIR USE GEORGETOWN UNIVERSITY (US) 2001-04-05 WO disclosed