SCHEMBL6990217

SCHEMBL6990217

CSc1ccc(-c2[nH]c(-c3ccccc3)c3c2CCCC3)cc1

nearest known ligand 0.87

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.47
PTGS1 P23219 1/20 0.47
HSD11B1 P28845 1/20 0.47
BRD4 O60885 1/20 0.44
CDKN1A P38936 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6998482 0.93 CDKN1A (0.44) PTGS2PTGS1BRD4CDKN1A
SCHEMBL6993952 0.84 HSD11B1 (0.59) HSD11B1BRD4
SCHEMBL6995905 0.83 PTGS2 (0.46) PTGS2PTGS1
SCHEMBL6992970 0.80 BRD4 (0.56) HSD11B1BRD4
SCHEMBL17283465 0.73 PTGS2 (0.63) PTGS2PTGS1
SCHEMBL403028 0.73 PTGS2 (0.63) PTGS2PTGS1
SCHEMBL8654013 0.73 PTGS2 (0.62) PTGS2PTGS1
SCHEMBL6991232 0.72 BRD4 (0.57) HSD11B1BRD4
SCHEMBL7567894 0.72 PTGS2 (0.53) PTGS2PTGS1
Hydrogen Sulfide SCHEMBL19086306 0.71 PTGS2 (0.61) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0921119-B1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-07-02 EP disclosed
US-6114360-A Pyrrole compounds ADIR ET COMPAGNIE (FR) 2000-09-05 US disclosed
US-6063804-A Pyrrole compounds ADIR ET COMPAGNIE (FR) 2000-05-16 US disclosed
EP-0921119-A1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-06-09 EP disclosed