SCHEMBL6998482

SCHEMBL6998482

CSc1ccc(-c2[nH]c(-c3ccc(SC)cc3)c3c2CCCC3)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CDKN1A P38936 1/20 0.44
KDM4E B2RXH2 1/20 0.40
USP2 O75604 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
PTGS2 P35354 3/20 0.40
NISCH Q9Y2I1 1/20 0.40
BRD4 O60885 1/20 0.38
PTGS1 P23219 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6990217 0.93 PTGS2 (0.47) CDKN1APTGS2BRD4PTGS1
SCHEMBL6991232 0.78 BRD4 (0.57) KDM4EUSP2HPGDBRD4
SCHEMBL6995905 0.75 PTGS2 (0.46) KDM4EHPGDPTGS2NISCHPTGS1
SCHEMBL6989278 0.74 PTGS1 (0.52) PTGS2BRD4PTGS1
SCHEMBL7000563 0.73 BRD4 (0.59) CDKN1AKDM4EHPGDBRD4
SCHEMBL6993952 0.73 HSD11B1 (0.59) BRD4
SCHEMBL11186325 0.69 PTGS2 (0.39) PTGS2NISCH
SCHEMBL6987934 0.69 PTGS1 (0.52) PTGS2BRD4PTGS1
SCHEMBL6992970 0.69 BRD4 (0.56) KDM4EHPGDBRD4
SCHEMBL10300271 0.68 ALDH1A1 (0.50) PTGS2NISCHPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0921119-B1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-07-02 EP disclosed
US-6114360-A Pyrrole compounds ADIR ET COMPAGNIE (FR) 2000-09-05 US disclosed
US-6063804-A Pyrrole compounds ADIR ET COMPAGNIE (FR) 2000-05-16 US disclosed
EP-0921119-A1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-06-09 EP disclosed