SCHEMBL7001648

SCHEMBL7001648

CCc1ccccc1N1CCC([C@@H]2Cc3c(ccc(OC)c3OC)[C@H](NC=O)O2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
USP2 O75604 2/20 0.38
HTT P42858 2/20 0.38
LMNA P02545 1/20 0.38
KDM4E B2RXH2 5/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
MAPT P10636 3/20 0.36
GAA P10253 2/20 0.36
POLB P06746 1/20 0.36
MAPK1 P28482 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
TSHR P16473 1/20 0.34
PARP1 P09874 1/20 0.34
HSD17B10 Q99714 2/20 0.33
RAB9A P51151 2/20 0.33
MALT1 Q9UDY8 1/20 0.33
MEN1 O00255 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27562876 0.83 PARP1 (0.34) ALDH1A1L3MBTL1HTTLMNAKDM4E
SCHEMBL7000445 0.83 ADRA2A (0.41) ALDH1A1L3MBTL1USP2HTTLMNA
SCHEMBL7001646 0.82 SIGMAR1 (0.41) ALDH1A1GAAHSD17B10ADRA1DADRA1A
SCHEMBL27412635 0.70 DRD1 (0.38) LMNAKDM4ESMN1; SMN2PARP1HPGD
SCHEMBL6993213 0.70 ACHE (0.46) POLBMEN1KMT2A
SCHEMBL6994737 0.70 ADRA2A (0.41) KDM4EMAPTHSD17B10MEN1KMT2A
Hydrochloric Acid SCHEMBL27410357 0.70 DRD1 (0.38) LMNAKDM4ESMN1; SMN2PARP1HPGD
SCHEMBL6988766 0.69 DRD1 (0.38) ALDH1A1HTTSMN1; SMN2GAATSHR
SCHEMBL6996299 0.69 DRD1 (0.40) L3MBTL1LMNAKDM4ESMN1; SMN2PARP1
SCHEMBL6988760 0.69 DRD1 (0.38) ALDH1A1HTTSMN1; SMN2GAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015446-B1 (4-PIPERIDINYL)-1H-2-BENZOPYRAN DERIVATIVES USEFUL AS ANTIPSYCHOTIC AGENTS AVENTIS PHARMA INC (US) 2003-04-02 EP claimed
US-6004982-A SIDE EFFECT REDUCTION; SCHIZOPHRENIA HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US claimed
EP-1015446-B1 (4-PIPERIDINYL)-1H-2-BENZOPYRAN DERIVATIVES USEFUL AS ANTIPSYCHOTIC AGENTS AVENTIS PHARMA INC (US) 2003-04-02 EP disclosed