SCHEMBL7000445

SCHEMBL7000445

CCc1ccccc1N1CCC([C@@H]2Cc3c(ccc(OC)c3OC)[C@H](CN)O2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.41
ADRA2B P18089 2/20 0.41
ADRA2C P18825 2/20 0.41
HTR2C P28335 2/20 0.41
SLC6A3 Q01959 2/20 0.41
DRD1 P21728 3/20 0.40
KDM4E B2RXH2 5/20 0.39
ALDH1A1 P00352 5/20 0.39
L3MBTL1 Q9Y468 3/20 0.39
USP2 O75604 2/20 0.39
HTT P42858 2/20 0.39
LMNA P02545 1/20 0.39
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
PARP1 P09874 1/20 0.35
GAA P10253 2/20 0.35
MAPT P10636 2/20 0.35
POLB P06746 1/20 0.35
MAPK1 P28482 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6994737 0.86 ADRA2A (0.41) ADRA2AADRA2BADRA2CHTR2CSLC6A3
SCHEMBL6998213 0.84 ADRA2A (0.45) ADRA2AADRA2BADRA2CHTR2CSLC6A3
SCHEMBL6998208 0.84 ADRA2A (0.45) ADRA2AADRA2BADRA2CHTR2CSLC6A3
SCHEMBL6998211 0.84 ADRA2A (0.45) ADRA2AADRA2BADRA2CHTR2CSLC6A3
SCHEMBL7001648 0.83 ALDH1A1 (0.38) KDM4EALDH1A1L3MBTL1USP2HTT
SCHEMBL6994578 0.82 ADRA2A (0.43) ADRA2AADRA2BADRA2CHTR2CSLC6A3
SCHEMBL6994580 0.82 ADRA2A (0.43) ADRA2AADRA2BADRA2CHTR2CSLC6A3
SCHEMBL6994586 0.82 ADRA2A (0.43) ADRA2AADRA2BADRA2CHTR2CSLC6A3
SCHEMBL6995343 0.82 ACHE (0.48) MEN1KMT2A
SCHEMBL6995337 0.82 ACHE (0.48) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015446-B1 (4-PIPERIDINYL)-1H-2-BENZOPYRAN DERIVATIVES USEFUL AS ANTIPSYCHOTIC AGENTS AVENTIS PHARMA INC (US) 2003-04-02 EP disclosed
US-6004982-A SIDE EFFECT REDUCTION; SCHIZOPHRENIA HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US disclosed