SCHEMBL7001664

SCHEMBL7001664

Nc1cc(-c2cccc(C(F)(F)F)c2)[nH]n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.60
IKBKB O14920 1/20 0.55
LMNA P02545 1/20 0.52
ALDH1A1 P00352 2/20 0.51
KMT2A Q03164 2/20 0.51
MITF O75030 1/20 0.51
TP53 P04637 1/20 0.51
SCN2A Q99250 2/20 0.51
NOTUM Q6P988 1/20 0.49
IDO1 P14902 1/20 0.49
MKNK1 Q9BUB5 1/20 0.47
MKNK2 Q9HBH9 1/20 0.47
MEN1 O00255 1/20 0.47
USP2 O75604 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
XDH P47989 1/20 0.47
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
NPY5R Q15761 1/20 0.45
ADORA2A P29274 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1854144 0.81 ALDH1A1 (0.70) KDRLMNAALDH1A1KMT2AMITF
SCHEMBL17413465 0.81 IKBKB (0.55) IKBKBKMT2ASCN2ANOTUMIDO1
SCHEMBL1853364 0.78 LMNA (0.56) LMNAALDH1A1KMT2AMITFTP53
SCHEMBL18284795 0.76 KDM4E (0.57) IKBKBLMNAALDH1A1KMT2ASCN2A
SCHEMBL330565 0.75 ALDH1A1 (0.66) LMNAALDH1A1KMT2AMITFTP53
SCHEMBL5068328 0.75 CYP1A2 (0.47) IKBKBSCN2ANOTUMIDO1
SCHEMBL6967479 0.75 MKNK1 (0.66) LMNAALDH1A1KMT2AMITFTP53
SCHEMBL6960706 0.75 ALDH1A1 (0.66) IKBKBLMNAALDH1A1KMT2AMITF
SCHEMBL28572920 0.75 SMN1; SMN2 (0.66) LMNAALDH1A1KMT2AMITFTP53
SCHEMBL30512092 0.75 SMN1; SMN2 (0.66) LMNAALDH1A1KMT2AMITFTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016001341-A1 SULFONYLAMINOPYRIDINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE F. HOFFMANN-LA ROCHE AG (CH) 2016-01-07 WO disclosed
EP-0945438-B1 PYRAZOLE DERIVATIVES BANYU PHARMA CO LTD (JP) 2003-03-05 EP disclosed
US-6057335-A Pyrazole derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 2000-05-02 US disclosed
EP-0945438-A1 PYRAZOLE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1999-09-29 EP disclosed