SCHEMBL17413465

SCHEMBL17413465

Cc1cc(-c2cccc(C(F)(F)F)c2)[nH]n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.55
NOTUM Q6P988 2/20 0.52
SCN2A Q99250 2/20 0.51
IDO1 P14902 1/20 0.49
MAPK14 Q16539 1/20 0.47
RAF1 P04049 1/20 0.46
NPY5R Q15761 1/20 0.45
BRD4 O60885 1/20 0.44
PIN1 Q13526 1/20 0.44
KDM1A O60341 1/20 0.44
CYP1A2 P05177 1/20 0.43
PIM1 P11309 2/20 0.43
MEN1 O00255 1/20 0.43
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43
EPHX2 P34913 1/20 0.43
MAP4K4 O95819 1/20 0.42
GPX4 P36969 1/20 0.42
GSK3B P49841 1/20 0.42
PIM3 Q86V86 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14616445 0.86 CTSS (0.50) IKBKBNOTUMSCN2AIDO1MAPK14
SCHEMBL19728985 0.85 KIF11 (0.49) IKBKBNOTUMSCN2AMEN1POLB
SCHEMBL3055345 0.81 TNIK (0.52) NOTUMSCN2ARAF1POLBKMT2A
SCHEMBL7001664 0.81 KDR (0.60) IKBKBNOTUMSCN2AIDO1NPY5R
SCHEMBL12948535 0.78 POLB (0.39) NOTUMPOLB
SCHEMBL20465066 0.78 NOTUM (0.51) NOTUMIDO1NPY5RCYP1A2POLB
SCHEMBL1773863 0.75 RAB9A (0.61) POLB
SCHEMBL20411744 0.75 TRPV3 (0.40) NOTUMRAF1POLB
SCHEMBL5068328 0.75 CYP1A2 (0.47) IKBKBNOTUMSCN2AIDO1CYP1A2
SCHEMBL1413881 0.75 KMT2A (0.54) IKBKBRAF1PIN1CYP1A2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1802373-A Pyrazoloisoquinoline derivatives as kinase inhibitors AVENTIS PHARMA INC (US) 2006-07-12 CN claimed
WO-2016001341-A1 SULFONYLAMINOPYRIDINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE F. HOFFMANN-LA ROCHE AG (CH) 2016-01-07 WO disclosed
CN-1802373-A Pyrazoloisoquinoline derivatives as kinase inhibitors AVENTIS PHARMA INC (US) 2006-07-12 CN disclosed