SCHEMBL5068328

SCHEMBL5068328

FC(F)(F)c1cccc(Cc2cc(-c3cccc(C(F)(F)F)c3)[nH]n2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
HTR2C P28335 2/20 0.46
HTR2B P41595 2/20 0.46
SCN2A Q99250 2/20 0.46
NOTUM Q6P988 1/20 0.44
IDO1 P14902 2/20 0.43
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
HTR2A P28223 1/20 0.43
POLB P06746 1/20 0.43
IKBKB O14920 1/20 0.43
DAO P14920 1/20 0.43
MPO P05164 1/20 0.43
TAAR1 Q96RJ0 1/20 0.42
AKR1B1 P15121 1/20 0.41
LTA4H P09960 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28775522 0.93 HTR2C (0.45) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1853783 0.80 MPO (0.50) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL14718571 0.76 DAO (0.53) HTR2CHTR2BHTR2ADAOAKR1B1
SCHEMBL28570388 0.75 ALDH1A1 (0.44) CYP1A2CYP2C9NOTUMIDO1POLB
SCHEMBL7001664 0.75 KDR (0.60) SCN2ANOTUMIDO1IKBKB
SCHEMBL17413465 0.75 IKBKB (0.55) CYP1A2SCN2ANOTUMIDO1POLB
SCHEMBL28114539 0.74 RAB9A (0.53) POLB
SCHEMBL3237564 0.73 TAAR1 (0.64) HTR2CHTR2BIDO1HTR2ADAO
SCHEMBL2128638 0.69 ALDH1A1 (0.50) HTR2CHTR2BIDO1HTR2ADAO
SCHEMBL30047602 0.69 ALDH1A1 (0.50) HTR2CHTR2BIDO1HTR2ADAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1925617-A1 HETEROCYCLIC COMPOUND, AND PRODUCTION PROCESS AND USE THEREOF ASKA Pharmaceutical Co., Ltd. (JP) 2008-05-28 EP disclosed