SCHEMBL7002194

SCHEMBL7002194

O=C1OCc2c(O)ccc(O)c21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 9/20 0.53
MAOB P27338 5/20 0.53
AURKB Q96GD4 2/20 0.46
KDR P35968 2/20 0.46
NUAK1 O60285 1/20 0.46
IGF1R P08069 1/20 0.46
MET P08581 1/20 0.46
PIM1 P11309 1/20 0.46
SRC P12931 1/20 0.46
AXL P30530 1/20 0.46
AKT1 P31749 1/20 0.46
NEK2 P51955 1/20 0.46
PLK1 P53350 1/20 0.46
PTK2 Q05397 1/20 0.46
PKN1 Q16512 1/20 0.46
NEK6 Q9HC98 1/20 0.46
ALK Q9UM73 1/20 0.46
MEN1 O00255 3/20 0.40
MAPT P10636 3/20 0.40
KMT2A Q03164 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12553463 0.84 MAOA (0.47) MAOAMAOBAURKBKDRNUAK1
SCHEMBL6998523 0.80 KDM4E (0.51) MAOAMAOBAURKBKDRNUAK1
SCHEMBL17264241 0.80 ALOX5 (0.44) MAOAMAOBAURKBKDRNUAK1
SCHEMBL7001855 0.72 MAPT (0.53) MAOAMAOBAURKBKDRMEN1
SCHEMBL29793269 0.72 MAOB (0.47) MAOAMAOBAURKBKDRNUAK1
SCHEMBL78594 0.72 MAOB (0.47) MAOAMAOBAURKBKDRNUAK1
5,7-Dihydroxy-4-Methylphthalide SCHEMBL3505368 0.72 NUAK1 (0.58) MAOAMAOBAURKBKDRNUAK1
SCHEMBL15680616 0.71 KDM4E (0.46) MAOAMAOBAURKBKDRNUAK1
SCHEMBL30487613 0.70 MAOA (1.00) MAOAMAOBAURKBKDRNUAK1
SCHEMBL20652853 0.69 MAOA (0.50) MAOAMAOBAURKBKDRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11731980-B1 Furo[3,4-b]quinolone compounds as antibacterial agents King Faisal University (SA) 2023-08-22 US disclosed
US-11731980-B1 Furo[3,4-b]quinolone compounds as antibacterial agents King Faisal University (SA) 2023-08-22 US disclosed
US-11731980-B1 Furo[3,4-b]quinolone compounds as antibacterial agents King Faisal University (SA) 2023-08-22 US disclosed
EP-1241169-B1 Isoindoloindolone derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-08-27 EP disclosed
US-6465660-B1 PARTICULARLY 2-HYDROXY-8,9-DIMETHOXYISOINDOLO(2,1-A)INDOL-6-ONE AND 2-HYDROXY-8,9-DIMETHOXYISOINDOLO(2,1-A)INDOL-6-ONE; TREATING A DISORDER OF THE MELATONINERGIC SYSTEM LES LABORATOIRES SERVIER (FR) 2002-10-15 US disclosed
EP-1241169-A1 Isoindoloindolone derivatives, process for their preparation and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2002-09-18 EP disclosed
US-5849750-A Dynemicin analogs CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 1998-12-15 US disclosed
US-5763451-A Dynemicin analogs CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 1998-06-09 US disclosed
WO-1996003124-A9 DYNEMICIN ANALOGS 1996-03-14 WO disclosed
WO-1996003124-A1 DYNEMICIN ANALOGS CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 1996-02-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11731980-B1 Furo[3,4-b]quinolone compounds as antibacterial agents TOP2A, TOP2B, TOP1 MAOA 770/4885MAOB 381/4885AURKB 363/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.