SCHEMBL7003424

SCHEMBL7003424

O=C(O)CN(CC(=O)O)Cc1c(-c2ccccc2)nc2ccccc2c1C(=O)NCCC1CCCCC1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.50
TACR3 P29371 15/20 0.47
TACR2 P21452 12/20 0.47
OPRM1 P35372 7/20 0.47
TP53 P04637 1/20 0.45
KCNH2 Q12809 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6625208 0.89 LMNA (0.53) LMNATACR3TACR2OPRM1TP53
SCHEMBL6626579 0.84 ALDH1A1 (0.56) LMNATACR3TACR2OPRM1TP53
SCHEMBL4667076 0.82 LMNA (0.48) LMNATACR3TACR2OPRM1TP53
SCHEMBL4665926 0.82 LMNA (0.48) LMNATACR3TACR2OPRM1TP53
SCHEMBL6629503 0.81 LMNA (0.52) LMNATACR3TACR2OPRM1TP53
SCHEMBL7096193 0.81 TACR3 (0.69) TACR3TACR2OPRM1KCNH2
SCHEMBL5908992 0.80 TACR3 (0.68) TACR3TACR2OPRM1
SCHEMBL5909008 0.80 TACR3 (0.68) TACR3TACR2OPRM1
SCHEMBL5042680 0.80 LMNA (0.47) LMNATACR3TACR2OPRM1TP53
SCHEMBL4665219 0.79 TACR3 (0.47) LMNATACR3TACR2OPRM1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1351953-A1 QUINOLINE DERIVATIVES AS NK-3 ANTAGONISTS GlaxoSmithKline S.p.A. (IT) 2003-10-15 EP disclosed
WO-2002044165-A1 QUINOLINE DERIVATIVES AS NK-3 ANTAGONISTS GLAXOSMITHKLINE SPA (IT) 2002-06-06 WO disclosed