SCHEMBL7007040

SCHEMBL7007040

CN(Cc1ccc(Cl)cc1)C(=O)c1n[nH]c2ncc(CN3CCOCC3)cc2c1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE1B Q01064 1/20 0.45
AKR1C3 P42330 1/20 0.44
NR1H4 Q96RI1 1/20 0.43
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
LSS P48449 1/20 0.41
F10 P00742 1/20 0.40
KCNH2 Q12809 3/20 0.40
POLA1 P09884 1/20 0.39
AURKA O14965 1/20 0.39
JAK2 O60674 1/20 0.39
JAK3 P52333 1/20 0.39
GSK3B P49841 1/20 0.39
DYRK1A Q13627 1/20 0.39
ENPP2 Q13822 1/20 0.39
HIF1A Q16665 1/20 0.38
EPAS1 Q99814 1/20 0.38
CHEK1 O14757 1/20 0.38
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6667774 0.87 CHEK1 (0.46) PDE1BAKR1C3NR1H4NPC1RAB9A
SCHEMBL6667470 0.83 INSR (0.39) AKR1C3NR1H4NPC1RAB9ALSS
SCHEMBL6667754 0.81 AKR1C3 (0.39) PDE1BAKR1C3NR1H4NPC1RAB9A
SCHEMBL7014636 0.81 RAB9A (0.38) NR1H4NPC1RAB9AF10ENPP2
SCHEMBL7015761 0.80 ALDH1A1 (0.41) NR1H4NPC1RAB9AF10SMN1; SMN2
SCHEMBL7478855 0.80 POLA1 (0.39) PDE1BAKR1C3NR1H4NPC1RAB9A
SCHEMBL7472513 0.79 AKR1C3 (0.36) PDE1BAKR1C3NR1H4NPC1RAB9A
SCHEMBL7014028 0.77 ALDH1A1 (0.37) NR1H4NPC1RAB9A
SCHEMBL7475511 0.77 NR1H4 (0.38) AKR1C3NR1H4NPC1RAB9ALSS
SCHEMBL6669285 0.76 POLA1 (0.35) AKR1C3NR1H4NPC1RAB9AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1301493-A2 HETEROCYCLE CARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2003-04-16 EP disclosed
WO-2002004444-A2 HETEROCYCLE CARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2002-01-17 WO disclosed