SCHEMBL7010649

SCHEMBL7010649

Cc1nn(Cc2ccc(C(=O)c3ccc(F)cc3)cc2)c2cnn(C(C)(C)C)c(=O)c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 4/20 0.46
PKLR P30613 3/20 0.46
RAB9A P51151 3/20 0.40
HTT P42858 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
MITF O75030 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
SCD O00767 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
NPC1 O15118 2/20 0.39
TP53 P04637 2/20 0.39
SLC2A1 P11166 1/20 0.39
TSHR P16473 1/20 0.39
HDAC3 O15379 2/20 0.38
HDAC4 P56524 2/20 0.38
HDAC1 Q13547 2/20 0.38
HDAC7 Q8WUI4 2/20 0.38
HDAC2 Q92769 2/20 0.38
HDAC10 Q969S8 2/20 0.38
HDAC11 Q96DB2 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7010994 0.91 ALDH1A1 (0.41) PKMPKLRRAB9AHTTMITF
SCHEMBL7010543 0.84 RAB9A (0.40) PKMRAB9AHTTNPSR1MITF
SCHEMBL7009974 0.82 PKM (0.45) PKMPKLRRAB9AHTTNPSR1
SCHEMBL7008568 0.77 PKM (0.41) PKMPKLRHTTMITFTDP1
SCHEMBL7015953 0.74 SMN1; SMN2 (0.41) PKMRAB9AHTTNPSR1MITF
SCHEMBL7012894 0.72 SMN1; SMN2 (0.48) PKMPKLRRAB9AHTTNPSR1
SCHEMBL9239206 0.71 MAPK14 (0.44) PKMRAB9AHTTNPSR1MITF
SCHEMBL9239707 0.71 RAB9A (0.67) PKMRAB9AHTTNPSR1MITF
SCHEMBL7015600 0.67 MAPT (0.43) TP53MAPTLMNAKDM4E
SCHEMBL7012827 0.65 TSHR (0.46) PKMPKLRRAB9AHTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed