SCHEMBL7012890

SCHEMBL7012890

Cn1c(SCc2ccc(C(=O)c3ccc(Cl)cc3)cc2)nc2[nH]ncc2c1=O

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 8/20 0.60
SMN1; SMN2 Q16637 2/20 0.52
MAPT P10636 3/20 0.51
THRB P10828 2/20 0.48
HTT P42858 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
RAB9A P51151 3/20 0.47
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
ALDH1A1 P00352 3/20 0.46
LMNA P02545 4/20 0.45
NPC1 O15118 2/20 0.42
RXFP1 Q9HBX9 1/20 0.42
ALDH1A2 O94788 1/20 0.42
ALDH1A3 P47895 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7010698 0.90 TP53 (0.51) TP53SMN1; SMN2MAPTTHRBHTT
SCHEMBL7016967 0.88 TP53 (0.58) TP53SMN1; SMN2MAPTTHRBHTT
SCHEMBL7017363 0.81 MAOA (0.46) TP53MAPTTHRBHTTMEN1
SCHEMBL7009666 0.80 MAOA (0.47) TP53SMN1; SMN2MAPTTHRBHTT
SCHEMBL7011002 0.80 MEN1 (0.48) TP53SMN1; SMN2MAPTTHRBHTT
SCHEMBL7011645 0.80 ALDH1A1 (0.58) TP53MAPTTHRBHTTMEN1
SCHEMBL7015339 0.80 KMT2A (0.68) TP53SMN1; SMN2MAPTTDP1MEN1
SCHEMBL7013210 0.80 MEN1 (0.53) TP53MAPTTHRBTDP1MEN1
SCHEMBL7016571 0.79 MAOA (0.54) TP53SMN1; SMN2MAPTTHRBHTT
SCHEMBL9060596 0.78 MAOA (0.52) TP53SMN1; SMN2MAPTTHRBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed