SCHEMBL7016967

SCHEMBL7016967

CCn1c(SCc2ccc(C(=O)c3ccc(Cl)cc3)cc2)nc2[nH]ncc2c1=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 7/20 0.58
KMT2A Q03164 3/20 0.52
ALDH1A1 P00352 3/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
MAPT P10636 4/20 0.49
THRB P10828 1/20 0.49
HTT P42858 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
LMNA P02545 3/20 0.46
MEN1 O00255 2/20 0.44
DRD2 P14416 3/20 0.43
TBXA2R P21731 3/20 0.43
KDM1A O60341 1/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7012890 0.88 TP53 (0.60) TP53KMT2AALDH1A1SMN1; SMN2MAPT
SCHEMBL7010698 0.78 TP53 (0.51) TP53KMT2AALDH1A1SMN1; SMN2MAPT
SCHEMBL7014540 0.74 DRD2 (0.52) TP53KMT2AALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL7013837 0.72 KMT2A (0.40) TP53KMT2AALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL7017363 0.71 MAOA (0.46) TP53KMT2AALDH1A1MAPTTHRB
SCHEMBL7012539 0.71 KMT2A (0.44) TP53KMT2AALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL7014308 0.71 DRD2 (0.59) TP53KMT2AALDH1A1MAPTMEN1
SCHEMBL7011645 0.71 ALDH1A1 (0.58) TP53KMT2AALDH1A1MAPTTHRB
SCHEMBL7016571 0.69 MAOA (0.54) TP53KMT2AALDH1A1SMN1; SMN2MAPT
Hydrochloric Acid SCHEMBL7012516 0.69 HRH3 (0.49) KMT2AALDH1A1SMN1; SMN2L3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed