SCHEMBL7016155

SCHEMBL7016155

Cn1c(=O)c2c(ccn2Cc2ccc(C(=O)c3ccc(Cl)nc3)cc2)n(C)c1=O

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 8/20 0.43
LMNA P02545 4/20 0.43
MAPK1 P28482 1/20 0.43
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.40
HTT P42858 2/20 0.40
UBE2N P61088 2/20 0.40
ABCC8 Q09428 1/20 0.39
KCNJ11 Q14654 1/20 0.39
ADORA2B P29275 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
GLA P06280 1/20 0.38
PPARG P37231 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7013633 0.87 LMNA (0.51) TRPA1LMNAMAPK1HTTMAOA
SCHEMBL7012643 0.83 TRPA1 (0.58) TRPA1RXFP1L3MBTL1MAPT
SCHEMBL7016345 0.83 LMNA (0.66) LMNAMAPK1SMN1; SMN2HTTUBE2N
SCHEMBL7009394 0.81 TRPA1 (0.61) TRPA1KDM4ESMN1; SMN2ABCC8KCNJ11
SCHEMBL7102075 0.80 KMT2A (0.46) LMNAMAPK1KDM4ESMN1; SMN2ADORA2B
SCHEMBL8644499 0.79 LMNA (0.51) LMNAMAPK1KDM4ESMN1; SMN2HTT
SCHEMBL7011108 0.71 LMNA (0.84) LMNAMAPK1SMN1; SMN2HTTUBE2N
Hydrochloric Acid SCHEMBL7019827 0.70 LMNA (0.82) LMNAMAPK1SMN1; SMN2HTTUBE2N
SCHEMBL8644491 0.70 RXFP1 (0.59) LMNAKDM4ESMN1; SMN2HTTADORA2B
Hydrochloric Acid SCHEMBL7013530 0.69 L3MBTL1 (0.39) LMNAKMT2AL3MBTL1PPARGMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed