SCHEMBL7102075

SCHEMBL7102075

Cn1c(=O)c2c(ccn2Cc2ccc(C(=O)c3ccc(N4CCN(c5ccccc5)CC4)nc3)cc2)n(C)c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.44
MEN1 O00255 4/20 0.42
ALDH1A1 P00352 5/20 0.42
HTR7 P34969 1/20 0.40
HTR6 P50406 1/20 0.40
MAPK8 P45983 2/20 0.39
TSHR P16473 3/20 0.39
ADORA2B P29275 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
MAPT P10636 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
USP2 O75604 2/20 0.39
MAPK1 P28482 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7016155 0.80 TRPA1 (0.43) KMT2AL3MBTL1ADORA2BSMN1; SMN2RXFP1
SCHEMBL7013633 0.76 LMNA (0.51) RAB9ATSHRMAPTMAPK1LMNA
SCHEMBL7012643 0.75 TRPA1 (0.58) L3MBTL1ALDH1A1RXFP1MAPT
SCHEMBL7015781 0.75 KMT2A (0.45) KMT2ANPC1RAB9AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL7017592 0.74 KMT2A (0.44) KMT2ANPC1RAB9AMEN1ALDH1A1
SCHEMBL7009394 0.72 TRPA1 (0.61) ALDH1A1SMN1; SMN2KDM4E
SCHEMBL7017996 0.70 LMNA (0.48) KMT2ARAB9AL3MBTL1MEN1ALDH1A1
SCHEMBL7015205 0.69 L3MBTL1 (0.57) RAB9AL3MBTL1ALDH1A1HTR7HTR6
Hydrochloric Acid SCHEMBL7018696 0.68 KMT2A (0.43) KMT2ANPC1RAB9AL3MBTL1MEN1
SCHEMBL7013690 0.68 KMT2A (0.47) KMT2ANPC1RAB9AL3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed