SCHEMBL7016471

SCHEMBL7016471

CC(=O)Oc1ccc(C(=O)c2ccc(CSc3nc4scc(C)c4c(=O)n3C)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 2/20 0.40
USP2 O75604 2/20 0.40
TSHR P16473 2/20 0.40
NPY1R P25929 1/20 0.40
NPY2R P49146 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
HTT P42858 3/20 0.39
ALDH1A1 P00352 2/20 0.39
PKM P14618 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
DAO P14920 1/20 0.39
POLB P06746 1/20 0.38
HSD17B10 Q99714 1/20 0.38
KDM4E B2RXH2 1/20 0.38
GFER P55789 1/20 0.38
MAPT P10636 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7012693 0.88 RXFP1 (0.42) TGM2USP2TSHRNPY1RNPY2R
SCHEMBL7018636 0.87 MAOA (0.46) TGM2USP2TSHRNPY1RNPY2R
SCHEMBL9051500 0.84 PSMB1 (0.50) ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL7018187 0.83 PSMB1 (0.49) KDM4E
SCHEMBL7017587 0.82 SMN1; SMN2 (0.44) ALDH1A1SMN1; SMN2KDM4EMAPTKMT2A
SCHEMBL7010770 0.82 MEN1 (0.47) RXFP1HTTALDH1A1PKMSMN1; SMN2
SCHEMBL7013586 0.80 SMN1; SMN2 (0.65) RXFP1HTTALDH1A1PKMSMN1; SMN2
SCHEMBL7011149 0.74 MEN1 (0.45) RXFP1HTTALDH1A1PKMSMN1; SMN2
SCHEMBL7013156 0.73 DAO (0.50) RXFP1HTTALDH1A1DAOPOLB
SCHEMBL7011506 0.72 MEN1 (0.55) USP2RXFP1HTTALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed