SCHEMBL7018636

SCHEMBL7018636

Cc1csc2nc(SCc3ccc(C(=O)c4ccc(Cl)cc4)cc3)n(C)c(=O)c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.46
MAOB P27338 1/20 0.46
LMNA P02545 1/20 0.43
RXFP1 Q9HBX9 1/20 0.41
TGM2 P21980 2/20 0.41
PKM P14618 2/20 0.41
HTT P42858 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
RAB9A P51151 1/20 0.41
ALDH1A1 P00352 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPT P10636 2/20 0.41
TP53 P04637 1/20 0.41
THRB P10828 1/20 0.41
KDM4E B2RXH2 2/20 0.40
ADRB2 P07550 1/20 0.40
GFER P55789 1/20 0.40
DRD2 P14416 1/20 0.40
TBXA2R P21731 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7012693 0.91 RXFP1 (0.42) RXFP1TGM2PKMHTTMEN1
SCHEMBL7016471 0.87 TGM2 (0.40) RXFP1TGM2PKMHTTMEN1
SCHEMBL7018169 0.84 KDM4E (0.57) MAOAMAOBLMNAHTTMEN1
SCHEMBL9051500 0.81 PSMB1 (0.50) ALDH1A1KDM4E
SCHEMBL7018370 0.81 MEN1 (0.50) MAOAMAOBLMNARXFP1PKM
SCHEMBL7011263 0.81 MAOA (0.52) MAOAMAOBLMNARXFP1HTT
Hydrochloric Acid SCHEMBL7018187 0.80 PSMB1 (0.49) KDM4E
SCHEMBL9060596 0.80 MAOA (0.52) MAOAMAOBLMNARXFP1PKM
SCHEMBL7017587 0.80 SMN1; SMN2 (0.44) LMNAKMT2ARAB9AALDH1A1SMN1; SMN2
SCHEMBL7019775 0.79 MEN1 (0.58) MAOAMAOBMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed