SCHEMBL7026352

SCHEMBL7026352

O=S(=O)(CCC=C(F)F)c1ccncc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.41
KMT2A Q03164 1/20 0.41
MMP1 P03956 2/20 0.38
RAB9A P51151 1/20 0.35
CLK1 P49759 2/20 0.34
CA2 P00918 3/20 0.33
NFE2L2 Q16236 2/20 0.33
KEAP1 Q14145 1/20 0.33
CYP3A4 P08684 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
CYP2D6 P10635 1/20 0.32
ALDH1A1 P00352 1/20 0.32
PAX8 Q06710 1/20 0.32
MAPK13 O15264 1/20 0.31
MAPK12 P53778 1/20 0.31
MAPK11 Q15759 1/20 0.31
MAPK14 Q16539 1/20 0.31
HSD11B1 P28845 1/20 0.31
NAMPT P43490 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4682707 0.74 CA2 (0.59) NPC1KMT2AMMP1RAB9ACLK1
SCHEMBL7023947 0.72 NFE2L2 (0.46) NPC1KMT2ARAB9ANFE2L2KEAP1
SCHEMBL4682702 0.71 NPC1 (0.50) NPC1KMT2AMMP1RAB9ACLK1
SCHEMBL4682791 0.71 CA2 (0.61) NPC1KMT2AMMP1CA2NFE2L2
SCHEMBL21693464 0.70 AOC3 (0.35) NPC1KMT2ARAB9AALDH1A1
SCHEMBL7023577 0.70 RAB9A (0.47) NPC1KMT2ARAB9ACYP3A4CYP2C9
SCHEMBL6096854 0.70 KMT2A (0.53) NPC1KMT2AMMP1RAB9ACYP3A4
SCHEMBL4681762 0.69 CA2 (0.62) NPC1KMT2AMMP1CA2NFE2L2
SCHEMBL8463226 0.69 FDPS (0.30)
Hydrochloric Acid SCHEMBL21646234 0.69 LOXL2 (0.36) NPC1KMT2ARAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749433-B1 (4,4-DIFLUOROBUT-3-ENYLTHIO)-SUBSTITUTED HETEROCYCLIC OR CARBOCYCLIC RING COMPOUNDS HAVING PESTICIDAL ACTIVITY SYNGENTA LTD (GB) 2003-05-07 EP disclosed
US-5952359-A NEMATICIDES, INSECTICIDES AND MITICIDES; 1,1-DIFLUORO-3-(THIAZOLYL OR ISOTHIAZOYL-THIO (OR SULFINYL OR SULFONYL)-PROP-1-ENE DERIVATIVES ZENECA LIMITED (GB) 1999-09-14 US disclosed
US-5912243-A NOVEL COMPOUNDS FOR CONTROLLING NEMATODES, INSECT OR ACARID PESTS ZENECA LIMITED (GB) 1999-06-15 US disclosed
US-5705516-A NEMATOCIDES, INSECTICIDES, ACARICIDES ZENECA LIMITED (GB) 1998-01-06 US disclosed
EP-0749433-A1 (4,4-DIFLUOROBUT-3-ENYLTHIO)-SUBSTITUTED HETEROCYCLIC OR CARBOCYCLIC RING COMPOUNDS HAVING PESTICIDAL ACTIVITY ZENECA LIMITED (GB) 1996-12-27 EP disclosed
WO-1995024403-A1 (4,4-DIFLUOROBUT-3-ENYLTHIO)-SUBSTITUTED HETEROCYCLIC OR CARBOCYCLIC RING COMPOUNDS HAVING PESTICIDAL ACTIVITY ZENECA LIMITED (GB) 1995-09-14 WO disclosed